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CAS No.: 1051375-16-6
Synonyms: S/GSK1349572;GSK1349572;Tivicay
Dolutegravir is an integrase inhibitor (IC50= 2.7 nM), modest activity against raltegravir-resistant signature mutants Y143R, Q148K, N155H, and G140S/Q148H.
生物活性
靶点 | HIV Integrase IC50:2.7nM |
动物研究 | ||||||||||||||||||||||||||||||||||
剂量 | Rat: ≤500 mg/kg[3] (p.o.) Monkey: 50 mg/kg - 500 mg/kg[3] (p.o.) | |||||||||||||||||||||||||||||||||
给药途径 | p.o. | |||||||||||||||||||||||||||||||||
动物药代数据 |
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NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT00867152 | Healthy Volunteer | Phase 1 | Completed | - | United States, New York ... more >> GSK Investigational Site Buffalo, New York, United States, 14202 Collapse << |
NCT00858455 | Healthy Volunteer | Phase 1 | Completed | - | United States, New York ... more >> GSK Investigational Site Buffalo, New York, United States, 14202 Collapse << |
NCT01302847 | HIV Infections | Phase 1 Phase 2 | Recruiting | June 30, 2023 | - |
实验方案
技术信息
CAS号 | 1051375-16-6 | 储存条件 |
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分子式 | C20H19F2N3O5 | 运输 | 蓝冰 | |||||||||||||
分子量 | 419.38 | 别名 | S/GSK1349572;GSK1349572;Tivicay;度鲁特韦 | |||||||||||||
溶解度 |
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动物实验配方 |
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Cell Lines | Concentration | Assay Type | Time | Activity Description | Data Sources |
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MDCK2 cells | - | Function assay | - | Inhibition of human OCT2 expressed in MDCK2 cells using [14C]metformin as substrate by liquid scintillation counting analysis | 23132334 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT00867152 | Healthy Volunteer | Phase 1 | Completed | - | United States, New York ... more >> GSK Investigational Site Buffalo, New York, United States, 14202 Collapse << |
NCT00858455 | Healthy Volunteer | Phase 1 | Completed | - | United States, New York ... more >> GSK Investigational Site Buffalo, New York, United States, 14202 Collapse << |
NCT01302847 | HIV Infections | Phase 1 Phase 2 | Recruiting | June 30, 2023 | - |
NCT01231542 | Infection, Human Immunodeficie... more >>ncy Virus Collapse << | Phase 1 | Completed | - | United States, Maryland ... more >> GSK Investigational Site Baltimore, Maryland, United States, 21287-5554 Collapse << |
NCT02178592 | Infection, Human Immunodeficie... more >>ncy Virus Collapse << | Phase 3 | Active, not recruiting | December 31, 2019 | - |
NCT02831673 | Infection, Human Immunodeficie... more >>ncy Virus Collapse << | Phase 3 | Active, not recruiting | March 3, 2020 | - |
NCT00708110 | Infection, Human Immunodeficie... more >>ncy Virus Collapse << | Phase 2 | Completed | - | United States, California ... more >> GSK Investigational Site Bakersfield, California, United States, 93301 GSK Investigational Site Long Beach, California, United States, 90813 GSK Investigational Site Newport Beach, California, United States, 92663 GSK Investigational Site Northridge, California, United States, 91325 GSK Investigational Site San Francisco, California, United States, 94115 United States, Colorado GSK Investigational Site Denver, Colorado, United States, 80220 United States, District of Columbia GSK Investigational Site Washington, District of Columbia, United States, 20009 United States, Florida GSK Investigational Site Fort Lauderdale, Florida, United States, 33316 GSK Investigational Site Ft. Lauderdale, Florida, United States, 33306 GSK Investigational Site Orlando, Florida, United States, 32803 GSK Investigational Site Vero Beach, Florida, United States, 32960 United States, Georgia GSK Investigational Site Atlanta, Georgia, United States, 30308 United States, New Jersey GSK Investigational Site Hillsborough, New Jersey, United States, 08844 GSK Investigational Site Voorhees, New Jersey, United States, 08043 United States, New Mexico GSK Investigational Site Santa Fe, New Mexico, United States, 87505 United States, North Carolina GSK Investigational Site Charlotte, North Carolina, United States, 28209 United States, Texas GSK Investigational Site Dallas, Texas, United States, 75204 GSK Investigational Site Dallas, Texas, United States, 75246 Collapse << |
NCT00708110 | - | - | Completed | - | - |
NCT03327740 | - | - | Active, not recruiting | June 30, 2019 | - |
NCT00828763 | Healthy Volunteer | Phase 1 | Completed | - | United States, Wisconsin ... more >> GSK Investigational Site Madison, Wisconsin, United States, 53704 Collapse << |
NCT00996021 | Healthy Subjects | Phase 1 | Completed | - | United States, Maryland ... more >> GSK Investigational Site Baltimore, Maryland, United States, 21225 Collapse << |
NCT00883935 | Healthy Volunteer | Phase 1 | Completed | - | United States, Texas ... more >> GSK Investigational Site Austin, Texas, United States, 78744 Collapse << |
NCT00774735 | Healthy Subjects ... more >> Infection, Human Immunodeficiency Virus Collapse << | Phase 1 | Completed | - | United States, New York ... more >> GSK Investigational Site Buffalo, New York, United States, 14202 Collapse << |
NCT03095638 | HIV Infections | Phase 1 | Completed | - | United States, Texas ... more >> GSK Investigational Site Austin, Texas, United States, 78744 Collapse << |
NCT00555035 | Healthy Subjects | Phase 1 | Completed | - | United States, Indiana ... more >> GSK Investigational Site Evansville, Indiana, United States, 47714 Collapse << |
NCT02486133 | HIV-Infection | Phase 3 | Active, not recruiting | December 2018 | Germany ... more >> Klinikum rechts der Isar Munich, Germany, 81675 Collapse << |
NCT02878642 | - | - | Recruiting | - | France ... more >> Caen University Hospital Recruiting Caen, France, 14000 Contact: Jean Jacques PARIENTI, MD, PhD parienti-jj@chu-caen.fr Collapse << |
NCT01622790 | Infection, Human Immunodeficie... more >>ncy Virus Collapse << | Phase 1 | Completed | - | United States, Kansas ... more >> GSK Investigational Site Overland Park, Kansas, United States, 66211 Collapse << |
NCT01332565 | Infection, Human Immunodeficie... more >>ncy Virus Collapse << | Phase 1 | Completed | - | United States, California ... more >> GSK Investigational Site Cypress, California, United States, 90630 Collapse << |
NCT00726336 | Healthy Subjects | Phase 1 | Completed | - | United States, New York ... more >> GSK Investigational Site Buffalo, New York, United States, 14202 Collapse << |
NCT02987530 | HIV-1 Infection | Phase 3 | Active, not recruiting | December 2019 | France ... more >> All The Regions Of The Country (40 Centers), France Collapse << |
NCT03360682 | HIV-1-infection ... more >> Solid Organ Transplant Collapse << | Phase 4 | Recruiting | January 2020 | Spain ... more >> Hospital Clínico y provincial de Barcelona Recruiting Barcelona, Spain, 08036 Contact: Anna Cruceta Arboles, MD +34 93 2275400 ext 4380 acruceta@clinic.ub.es Collapse << |
NCT01449929 | Infection, Human Immunodeficie... more >>ncy Virus Collapse << | Phase 3 | Completed | - | - |
NCT01231529 | Healthy Subjects ... more >> Hepatic Impairment Infection, Human Immunodeficiency Virus Collapse << | Phase 1 | Completed | - | United States, Minnesota ... more >> GSK Investigational Site Minneapolis, Minnesota, United States, 55404 Collapse << |
NCT01449929 | - | - | Completed | - | - |
NCT01536873 | Infection, Human Immunodeficie... more >>ncy Virus Collapse << | Phase 3 | Recruiting | August 2018 | - |
NCT03760458 | HIV Infections | Phase 1 Phase 2 | Not yet recruiting | August 2023 | United States, Illinois ... more >> Lurie Children's Hospital of Chicago (LCH) CRS Not yet recruiting Chicago, Illinois, United States, 60614-3393 Contact: Margaret Ann Sanders, M.P.H. 312-227-8275 msanders@luriechildrens.org Collapse << |
NCT01209065 | Infections, Human Immunodefici... more >>ency Virus and Herpesviridae Collapse << | Phase 1 | Completed | - | United States, New York ... more >> GSK Investigational Site Buffalo, New York, United States, 14202 Collapse << |
NCT03078556 | Infection, Human Immunodeficie... more >>ncy Virus Collapse << | Phase 1 | Completed | - | United States, Kansas ... more >> GSK Investigational Site Overland Park, Kansas, United States, 66211 Collapse << |
NCT02893488 | Infection, Human Immunodeficie... more >>ncy Virus Collapse << | Phase 1 | Completed | - | United States, Kansas ... more >> GSK Investigational Site Overland Park, Kansas, United States, 66211 Collapse << |
NCT03198884 | - | - | Active, not recruiting | May 1, 2018 | - |
NCT03683524 | HIV-1 Infection | Phase 4 | Not yet recruiting | October 2020 | - |
NCT01098526 | Infections, Human Immunodefici... more >>ency Virus and Herpesviridae Collapse << | Phase 1 | Completed | - | United States, New York ... more >> GSK Investigational Site Buffalo, New York, United States, 14202 Collapse << |
NCT01404806 | Healthy Adult Females | Phase 1 | Completed | - | United States, North Carolina ... more >> University of North Carolina, Chapel Hill Chapel Hill, North Carolina, United States, 27599 Collapse << |
NCT02370979 | HIV-1 Infection | Phase 4 | Unknown | July 2017 | France ... more >> Centre hospitalier de Belfort-Montbéliard Active, not recruiting Belfort, France, 90000 Centre hospitalier de Colmar Recruiting Colmar, France, 68024 Contact: Martin MARTINOT, MD martin.martinot@ch-colmar.fr Centre hospitalier de Mulhouse Recruiting Mulhouse Cedex, France, 68070 Contact: Geneviève BECK WIRTH, MD beck-wirthg@ch-mulhouse.fr Hôpitaux Universitaire de Strasbourg Recruiting Strasbourg Cedex, France, 67091 Contact: David REY, PhD david.rey@chru-strasbourg.fr Collapse << |
NCT02384395 | HIV Acute HIV... more >> Infection Collapse << | Not Applicable | Recruiting | July 2021 | United States, North Carolina ... more >> University of North Carolina Recruiting Chapel Hill, North Carolina, United States, 27599 Duke University Health System Recruiting Durham, North Carolina, United States, 27710 Contact: Kara McGee, MSPH, PA-C 919-668-0242 kara.mcgee@duke.edu Principal Investigator: Mehri McKellar, MD Collapse << |
NCT02513147 | HIV-1 | Phase 4 | Completed | - | Spain ... more >> Hospital Universitari Vall d'Hebron Barcelona, Spain, 08035 Collapse << |
NCT02738931 | Infection, Human Immunodeficie... more >>ncy Virus Collapse << | Phase 1 | Completed | - | United States, Kansas ... more >> GSK Investigational Site Overland Park, Kansas, United States, 66211 Collapse << |
NCT00774111 | Healthy Subjects | Phase 1 | Completed | - | United States, New York ... more >> GSK Investigational Site Buffalo, New York, United States, 14202 Collapse << |
NCT00631592 | Healthy Subjects | Phase 1 | Completed | - | United States, Wisconsin ... more >> GSK Investigational Site Madison, Wisconsin, United States, 53704 Collapse << |
NCT01366547 | Healthy Subjects ... more >> Infection, Human Immunodeficiency Virus Collapse << | Phase 1 | Completed | - | United States, New York ... more >> GSK Investigational Site Buffalo, New York, United States, 14202 Collapse << |
NCT01762995 | Infection, Human Immunodeficie... more >>ncy Virus Collapse << | Phase 1 | Completed | - | - |
NCT02777229 | HIV-1 Infection | Phase 3 | Active, not recruiting | July 2018 | Cameroon ... more >> Cité verte Hospital Yaoundé, Cameroon Hopital Central Yaoundé, Cameroon Military Hospital Yaoundé, Cameroon Collapse << |
NCT00950859 | Infection, Human Immunodeficie... more >>ncy Virus Collapse << | Phase 2 | Completed | - | - |
NCT02069834 | HIV Infection ... more >> HAART-treated Virologically Controlled Collapse << | Phase 2 Phase 3 | Withdrawn(One of the both Fund... more >>er partners decided to stop the study before the initiation thus no product provided and no funding to realize the study) Collapse << | October 2017 | France ... more >> CHU Guadeloupe Point-a-pitre, Guadeloupe, France, 97159 CHU de Fort de France Fort de France, Martinique, France, 87261 Chu Jean Minjoz Besançon, France, 25030 Hôpital Avicenne Bobigny, France, 93000 Hôpital Jean Verdier Bondy, France, 93140 CHU de Bordeaux Bordeaux, France, 33076 CHU de DIJON Dijon, France, 21079 CHD La Roche sur Yon La Roche sur Yon, France, 85925 CHU Kremlin Bicêtre Le Kremlin Bicetre, France, 94275 Hôpital Perpetuel Secours Levallois-perret, France, 92300 CHU de Nantes Nantes, France, 44093 Hôpital Saint Louis Paris Cedex 10, France, 75475 CHU BICHAT - Claude Bernard Paris cedex 18, France, 75877 CHU Hôtel Dieu Paris Paris, France, 75004 Hôpital La Pitié Salpêtrière Paris, France, 75013 Hôpital Necker - enfants Malades Paris, France, 75015 Hôpital Européen Georges Pompidou Paris, France, 75908 CHU de Rennes - Hôpital Pontchaillou Rennes, France, 35000 CH Delafontaine Saint Denis, France, 93200 CHU Saint Etienne Saint Etienne, France, 42055 CHU de Strasbourg Strasbourg, France, 67091 Hôpital FOCH Suresnes, France, 92150 CHU Toulouse Toulouse, France, 31059 CHRU de Tours Tours Cedex 09, France, 37044 CHU de Nancy VANDOEUVRE LES NANCY cedex, France, 54511 Collapse << |
NCT02064374 | Infection, Human Immunodeficie... more >>ncy Virus Collapse << | Phase 1 | Completed | - | United States, Kansas ... more >> GSK Investigational Site Overland Park, Kansas, United States, 66211 Collapse << |
NCT02656511 | HIV | Phase 4 | Recruiting | April 2020 | United States, California ... more >> San Francisco General Hospital Recruiting San Francisco, California, United States, 94110 Contact: Sulggi A Lee, MD PhD Sulggi.Lee@ucsf.edu Contact: Steven G Deeks, MD Steven.Deeks@ucsf.edu Collapse << |
NCT02337322 | Acquired Immune Deficiency Syn... more >>drome Virus Collapse << | Phase 4 | Active, not recruiting | December 2019 | Spain ... more >> Hospital Clinic of Barcelona Barcelona, BCN, Spain, 08013 Collapse << |
NCT00950859 | - | - | Completed | - | - |
NCT02582684 | HIV-1 Infection | Phase 2 | Completed | - | - |
NCT01098513 | Infection, Human Immunodeficie... more >>ncy Virus Collapse << | Phase 1 | Completed | - | United States, Texas ... more >> GSK Investigational Site Austin, Texas, United States, 78744 Collapse << |
NCT02715479 | Infection, Human Immunodeficie... more >>ncy Virus Collapse << | Phase 1 | Completed | - | United States, Texas ... more >> GSK Investigational Site Austin, Texas, United States, 78744 Collapse << |
NCT01827540 | HIV-infection/AIDS | Phase 1 | Completed | - | United States, Florida ... more >> SeaView Research, Inc. Miami, Florida, United States, 33126 Collapse << |
NCT02582684 | - | - | Completed | - | - |
NCT01382238 | Infections, Human Immunodefici... more >>ency Virus and Herpesviridae Collapse << | Phase 1 | Completed | - | United States, Texas ... more >> GSK Investigational Site Austin, Texas, United States, 78744 Collapse << |
NCT02659761 | Human Immunodeficiency Virus | Phase 4 | Recruiting | March 2019 | Ireland ... more >> Mater Misericordiae University Hospital Recruiting Dublin, Ireland, 7 Contact: Willard Tinago, PhD wtinago@gmail.com Contact: Patrick WG Mallon, MB BCh, PhD, FRCPI paddy.mallon@ucd.ie Principal Investigator: Patrick Mallon, MB BCh, PhD, FRCPI Sub-Investigator: Gerard Sheehan, MB BCh BAO, FRCPI Sub-Investigator: John Lambert, MD, PhD Collapse << |
NCT03017872 | HIV Infections | Phase 4 | Recruiting | December 28, 2021 | Argentina ... more >> Hospital G de Agudos JM Ramos Mejia Not yet recruiting Buenos Aires, Ciudad De Buenos Aires, Argentina, C1221ADC Contact: Marcelo Losso 5411 4127 0276 mlosso@hivramos.org.ar Contact: Guillermo Viloria 5411 4931 5252 gviloria@hivramos.org.ar Principal Investigator: Marcelo Losso, M.D. Hospital Dr Diego Paroissien Not yet recruiting Isidro Casanova, Provincia De Buenos Aires, Argentina, 1765 Contact: Eduardo Warley 5411 1541 897 181 eduwarley@yahoo.com.ar Contact: Maria Ines Vieni 5411 1136 877 377 ext 3340 inesvieni@gmail.com Principal Investigator: Eduardo Warley, M.D. CAICI Not yet recruiting Rosario, Provincia De Santa Fe, Argentina, S2000PBJ Contact: Sergio Lupo 54 9 341 515 7704 drsergiolupo@gmail.com Contact: Luciana Peroni 54 341 424 8045 administracioncaici@gmail.com Principal Investigator: Sergio Lupo, M.D. Hospital Interzonal de Agudos San Juan de Dios Recruiting La Plata, Argentina, 1900 Contact: Martha Michaan +54 9221 5765 131 mgmichaan@yahoo.com.ar Principal Investigator: Martha Michaan, M.D. Brazil Laboratório de Pesquisa Clinica Em Hiv/Aids - Instituto Nacional de Infectologia - Fiocruz Not yet recruiting Rio de Janeiro, Brazil, 21040-360 Contact: Beatriz Grinsztejn +552122707064 beatriz.grinsztejn@gmail.com Contact: Kelly Gama +552138659614 kelly.gama@ini.fiocruz.br Principal Investigator: Beatriz Grinsztejn, MD, PhD Chile Hospital San Borja-Arriaran Not yet recruiting Santiago, Chile, 8360159 Contact: Marcelo Wolff 562- 555 6206 marcewolff@yahoo.com Contact: Gladys Allendes 562-555-6206 gladys_allendes@yahoo.es Principal Investigator: Marcelo Wolff, MD Colombia ASISTENCIA Cientifica De Alta Complejidad S.A.S. Not yet recruiting Bogota, Colombia, 110010 Contact: Otto Sussmann 57-1- 5107600 ext 104 osussmann@gmail.com Contact: Ana Julia Rojas 57-1-5107600 ext 128 coord.investigaciones@asistenciacientifica.com Principal Investigator: Otto Sussmann, M.D. Guinea Centre de traitementambulatoire de Donka ( Hopital de jour) Not yet recruiting Conakry, Guinea, BP:5845 Contact: Mohamed Cisse +224 622 292 590 cissebibi1@gmail.com Contact: Thierno Mamadou Tounkara +224 622 318 171 tounkm@yahoo.fr Principal Investigator: Mohamed Cisse, Prof. India YRG Care Not yet recruiting Chennai, Tamil Nadu, India, 600113 Contact: Nagalingeswaran Kumarasamy 91 917 691 2007 kumarasamy@yrgcare.org Contact: Faith Beulah 91 44 39106811 beulah@yrgcare.org Principal Investigator: Nagalingeswaran Kumarasamy, MD Malaysia University of Malaya Medical Centre Recruiting Kuala Lumpur, Malaysia, 59100 Contact: Raja Iskandar Shah Raja Azwa 603-79493834 iskandar.azwa@gmail.com Contact: Margaret Tan 603-79492622 margarettan455@gmail.com Principal Investigator: Raja Iskandar Shah Raja Azwa, MBChB, MRCP Mali University of Sciences, Techniques and Technologies of Mali, University Clinical Research Center (UCRC) Not yet recruiting Bamako, Mali Contact: Sounkalo Doa +223 72274971 sounkalod@icermali.org Contact: Yacouba Cissoko +22374567649 or +22397195994 ycissoko@hotmail.com Principal Investigator: Sounkalo Doa, Prof. Mexico Morales Vargas Centro de Investigacion SC Not yet recruiting León, Guanajuato, Mexico, 37000 Contact: Juan Luis Mosqueda Gomez +52 (477) 1310037 luis_mosqueda@yahoo.com Contact: Jorge Morales Vargas +52 (477) 7160714 mnc.jorge@hotmail.com Hospital Civil de Guadalajara Not yet recruiting Guadalajara, Jalisco, Mexico, 44280 Contact: Jaime Andrade-Villanueva jandradev@msn.com Contact: Angeles González-Hernández 5233 3614 7586 angelesghdez1@gmail.com Principal Investigator: Jaime Andrade-Villanueva, M.D. Instituto Nacional de Ciencias Medicas y Nutriciòn Salvador Zubiran Not yet recruiting Mexico City, Mexico, 14080 Contact: Juan Sierra Madero 52 5556559675 jsmadero@yahoo.com Contact: Izchel Loyo iz.inncm@outlook.com Principal Investigator: Juan Sierra Madero, M.D. Nigeria Institute of Human Virology, Nigeria (IHVN) Not yet recruiting Abuja, Nigeria, 9396 Contact: Ernest Ekong +2348023107612 ernestekong@ihvnigeria.org Contact: Nnakelu Eriobu +2347039469273 neriobu@ihvnigeria.org Principal Investigator: Ernest Ekong, MD South Africa Desmond Tutu HIV Foundation Recruiting Cape Town, South Africa, 7925 Contact: Richard Kaplan Richard.Kaplan@hiv-research.org.za Contact: Christie Heiberg 27 21 406 3621 Christie.Heiberg@hiv-research.org.za Principal Investigator: Richard Kaplan, M.D. Clinical HIV Research Unit (CHRU), Wits Health Consotium (Pty) Ltd Recruiting Johannesburg, South Africa, 2041 Contact: Noluthando Mwelase tmwelase@witshealth.co.za Contact: Pauline Vunandala 27 11 276 8800 pvunandlala@witshealth.co.za Principal Investigator: Noluthando Mwelase, MBCHB Perinatal HIV Research Unit (PHRU), Chris Hani Baragwanath Hospital Recruiting Soweto, South Africa, 1864 Contact: Lerato Mohapi mohapil@hivsa.com Contact: Debra Peters 27 11 989 9700 petersd@phru.co.za Principal Investigator: Lerato Mohapi, BSc, MBBCh Thailand HIV-NAT (The HIV Netherlands Australia Thailand Research Collaboration), Thai Red Cross AIDS Research Centre Recruiting Bangkok, Thailand, 10330 Contact: Anchalee Avihingsanon +662 652 3040 ext 107 anchaleea2009@gmail.com Contact: Kanitta Pussadee +662 652 3040 ext 202 kanitta.p@hivnat.org Principal Investigator: Anchalee Avihingsanon, M.D. Chiangrai Prachanukroh Hospital Not yet recruiting Chiang Rai, Thailand, 57000 Contact: Pacharee Kantipong 66818859195 pachareek@hotmail.com Contact: Supawadee Pongprapass 66819616900 npudit@hotmail.com Principal Investigator: Pacharee Kantipong, M.D. Srinagarind Hospital, Khon Kaen University Recruiting Khon Kaen, Thailand, 40002 Contact: Ploenchan Chetchotisakd 6643363168 ploencha@kku.ac.th Contact: Anchalee Tiyabut 6643363169 atiyabut@yahoo.com Principal Investigator: Ploenchan Chetchotisakd, M.D. Bamrasnaradura Infectious Diseases Institute Recruiting Nonthaburi, Thailand, 11000 Contact: Weerawat Manosuthi drweerawat@hotmail.com Contact: Supeda Thongyen 6625903631 supeda_t@yahoo.com Principal Investigator: Weerawat Manosuthi, M.D. Zimbabwe University of Zimbabwe Clinical Research Centre Recruiting Harare, Zimbabwe, +263 Contact: James G Hakim 263 772225489 Jhakim@mweb.co.zw Contact: Shepherd Mudzingwa 263 4 701717 smudzingwa@yahoo.com Principal Investigator: James G Hakim, M.D. Collapse << |
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NCT02219217 | HIV | Phase 1 | Completed | - | United Kingdom ... more >> St Stephen's AIDS Trust London, United Kingdom, SW10 9NH Collapse << |
NCT02185300 | Infection, Human Immunodeficie... more >>ncy Virus Collapse << | Phase 1 | Completed | - | United States, Kansas ... more >> GSK Investigational Site Overland Park, Kansas, United States, 66211 Collapse << |
NCT02218320 | - | - | Completed | - | United States, North Carolina ... more >> Clinical and Translational Research Center, UNC Hospitals Chapel Hill, North Carolina, United States, 27599 Collapse << |
NCT02218320 | - | - | Completed | - | - |
NCT02211690 | Human Immunodeficiency Virus | Phase 4 | Completed | - | Australia, New South Wales ... more >> St Vincent's Hospital Centre for Applied Medical Research Darlinghurst, New South Wales, Australia, 2010 Sydney Sexual Health Centre Sydney, New South Wales, Australia, 2000 Clinic 16, Royal North Shore Hospital Sydney, New South Wales, Australia, 2065 Australia, Victoria Melbourne Sexual Health Centre Carlton, Victoria, Australia, 3053 Alfred Hospital Melbourne, Victoria, Australia, 3004 Collapse << |
NCT02542852 | HIV-1 Infection | Phase 2 | Recruiting | December 2017 | Italy ... more >> Ospedale San Raffaele Scientific Institute Recruiting Milan, Italy, 20127 Collapse << |
NCT03336346 | - | - | Recruiting | December 2018 | Botswana ... more >> Botswana-UPenn Partnership Recruiting Gaborone, Botswana Contact: Chelsea Morroni, MD 26776524112 chelseaamorroni@gmail.com Principal Investigator: Chelsea Morroni, MD Collapse << |
NCT02067767 | HIV-1 Infection | Phase 2 | Completed | - | France ... more >> La Roche-sur-Yon Hospital La Roche-sur-Yon, France Nantes University Hospital Nantes, France Collapse << |
NCT02499978 | HIV/AIDS | Phase 2 Phase 3 | Withdrawn | - | United States, California ... more >> Stanford Univerity Stanford, California, United States, 94305 United States, Colorado University of Colorado Aurora, Colorado, United States, 80045 Collapse << |
NCT01467531 | Infections, Human Immunodefici... more >>ency Virus and Hepatitis Collapse << | Phase 1 | Completed | - | United States, New York ... more >> GSK Investigational Site Buffalo, New York, United States, 14202 Collapse << |
NCT02242799 | Malaria HIV | Phase 1 | Completed | - | Uganda ... more >> Infectious Diseases Institute Kampala, Uganda Collapse << |
NCT03033836 | HIV Infections | Phase 4 | Active, not recruiting | July 2019 | Argentina ... more >> Fundacion Huesped Ciudad de Buenos Aires, Buenos Aires, Argentina, C1202ABB Collapse << |
NCT01966822 | HIV-1 Infection | Phase 3 | Completed | - | Spain ... more >> GermansTrias i Pujol Hospital Badalona, Barcelona, Spain, 08916 Hospital de la Santa Creu i Sant Pau Barcelona, Spain, 08025 Hospital Clínico San Carlos Madrid, Spain, 28040 Collapse << |
NCT03493568 | HIV-1-infection | Phase 3 | Recruiting | July 31, 2020 | Italy ... more >> Ospedale San Raffaele Recruiting Milan, Lombardia, Italy, 20127 Contact: ADRIANO LAZZARIN 0226437939 lazzarin.adriano@hsr.it Contact: Elisabetta Carini 0226437934 carini.elisabetta@hsr.it Ospedale San Raffaele Scientific Institute Recruiting Milan, Italy, 20127 Collapse << |
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NCT02596334 | HIV | Phase 3 | Terminated(5 patients on tivic... more >>ay had virological failure) Collapse << | - | France ... more >> CHD de VENDEE La Roche sur Yon, France, 85925 CH de LA ROCHELLE La Rochelle, France, 17019 CHRU de NANTES Nantes, France, 44093 CH de NIORT Niort, France, 79021 CHR d'ORLEANS Orleans, France, 45032 CHRU de POITIERS Poitiers, France, 86021 CHU de STRASBOURG Strasbourg, France, 67000 CHRU de TOURS Tours, France, 37044 CHU de NANCY Vandoeuvre Les Nancy, France, 54511 Collapse << |
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NCT01499199 | - | - | Completed | - | - |
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NCT02263326 | HIV Infection | Phase 3 | Completed | - | United States, California ... more >> University of California San Diego San Diego, California, United States United States, Georgia Emory University Atlanta, Georgia, United States United States, Illinois Northwestern University Chicago, Illinois, United States, 60611 United States, Massachusetts Brigham and Women's Hospital Boston, Massachusetts, United States United States, New York Cornell University New York, New York, United States United States, Ohio University of Cincinnati Cincinnati, Ohio, United States The Ohio State University Columbus, Ohio, United States Collapse << |
NCT03249181 | HIV-1-infection ... more >> Pregnancy Related Collapse << | Phase 3 | Active, not recruiting | March 2021 | South Africa ... more >> University of Cape Town Cape Town, Western Cape, South Africa Uganda Infectious Diseases Institute Kampala, Uganda Collapse << |
NCT01459315 | Healthy | Phase 1 | Completed | - | United States, North Carolina ... more >> University of North Carolina, Chapel Hill Chapel Hill, North Carolina, United States, 27599 Collapse << |
NCT02527096 | HIV-1 Infection | Phase 2 | Completed | - | France ... more >> Hôpital Avicenne Bobigny, France, 93009 Hôpital Saint-André Bordeaux, France, 33000 Hôpital Gabriel Montpied Clermont-Ferrand, France, 63003 Hôpital du Bocage Dijon, France, 21079 Hôpital Pierre Zobda-Quitman Fort de France, France, 97261 Hôpial Bicêtre Le Kremelin Bicêtre, France, 94270 Hôpital Gui de Chaudiac Montpellier, France, 34295 Hôpital de l'Hotel Dieu Nantes, France, 44093 Hôpital Saint-Louis Paris, France, 75010 Hôpital Saint-Antoine Paris, France, 75012 Hôpital Pitié-Salpêtrière Paris, France, 75013 Hôpital Necker Paris, France, 75015 Hôpital Bichat Paris, France, 75018 Centre hospitalier de Pernignan Perpignan, France, 66046 Hôpital Pontchaillou Rennes, France, 35033 Hôpital Purpan Toulouse, France, 31059 Hôpital Gustave Dron Tourcoing, France, 59208 Hôpital Bretonneau Tours, France, 37044 Collapse << |
NCT03602690 | HIV/AIDS | Phase 2 | Recruiting | October 3, 2020 | Cambodia ... more >> NCHADS Recruiting Phnom Penh, Cambodia Contact: Sun Ly Penh, MD Collapse << |
NCT02263326 | - | - | Completed | - | - |
NCT01353716 | Infection, Human Immunodeficie... more >>ncy Virus Collapse << | Phase 1 | Completed | - | United States, Minnesota ... more >> GSK Investigational Site Minneapolis, Minnesota, United States, 55404 Collapse << |
NCT01328041 | Infection, Human Immunodeficie... more >>ncy Virus Collapse << | Phase 3 | Completed | - | - |
NCT02285374 | HIV | Phase 4 | Unknown | December 2015 | United Kingdom ... more >> Chelsea and Westminster Hospital London, United Kingdom, SW10 9TH Collapse << |
NCT01498861 | Infection, Human Immunodeficie... more >>ncy Virus Collapse << | Phase 1 | Completed | - | United States, Florida ... more >> GSK Investigational Site Miami, Florida, United States, 33169 Collapse << |
NCT01328041 | - | - | Completed | - | - |
NCT03199690 | HIV-1-infection ... more >> Tuberculosis Collapse << | Phase 1 | Not yet recruiting | March 2018 | - |
NCT02551523 | Monotherapy D... more >>olutegravir Primary HIV Infection Treatment Efficacy Collapse << | Phase 2 | Active, not recruiting | February 2021 | Switzerland ... more >> University Hospital Zurich, University of Zurich Zurich, Switzerland, 8091 Collapse << |
NCT02245022 | HIV Pregnancy | Phase 2 Phase 3 | Active, not recruiting | December 2018 | South Africa ... more >> Desmond Tutu HIV Foundation Cape Town, Western Cape, South Africa Uganda Infectious Diseases Institute Kampala, Uganda Collapse << |
NCT02076386 | - | - | Completed | - | Germany ... more >> GSK Investigational Site Freiburg, Baden-Wuerttemberg, Germany, 79106 GSK Investigational Site Mannheim, Baden-Wuerttemberg, Germany, 68161 GSK Investigational Site Stuttgart, Baden-Wuerttemberg, Germany, 70197 GSK Investigational Site Tuebingen, Baden-Wuerttemberg, Germany, 72076 GSK Investigational Site Fuerth, Bayern, Germany, 90762 GSK Investigational Site Muenchen, Bayern, Germany, 80331 GSK Investigational Site Muenchen, Bayern, Germany, 80335 GSK Investigational Site Muenchen, Bayern, Germany, 80336 GSK Investigational Site Muenchen, Bayern, Germany, 80801 GSK Investigational Site Muenchen, Bayern, Germany, 81675 GSK Investigational Site Frankfurt am Main, Hessen, Germany, 60590 GSK Investigational Site Frankfurt, Hessen, Germany, 60311 GSK Investigational Site Hannover, Niedersachsen, Germany, 30159 GSK Investigational Site Osnabrueck, Niedersachsen, Germany, 49090 GSK Investigational Site Aachen, Nordrhein-Westfalen, Germany, 52062 GSK Investigational Site Bochum, Nordrhein-Westfalen, Germany, 44787 GSK Investigational Site Dortmund, Nordrhein-Westfalen, Germany, 44137 GSK Investigational Site Duesseldorf, Nordrhein-Westfalen, Germany, 40237 GSK Investigational Site Koeln, Nordrhein-Westfalen, Germany, 50674 GSK Investigational Site Muenster, Nordrhein-Westfalen, Germany, 48143 GSK Investigational Site Koblenz, Rheinland-Pfalz, Germany, 56073 GSK Investigational Site Mainz, Rheinland-Pfalz, Germany, 55116 GSK Investigational Site Magdeburg, Sachsen-Anhalt, Germany, 39120 GSK Investigational Site Berlin, Germany, 10243 GSK Investigational Site Berlin, Germany, 10405 GSK Investigational Site Berlin, Germany, 10439 GSK Investigational Site Berlin, Germany, 10707 GSK Investigational Site Berlin, Germany, 10777 GSK Investigational Site Berlin, Germany, 10961 GSK Investigational Site Berlin, Germany, 13347 GSK Investigational Site Berlin, Germany, 14057 GSK Investigational Site Chemnitz, Germany, 09111 GSK Investigational Site Hamburg, Germany, 20099 GSK Investigational Site Hamburg, Germany, 20146 GSK Investigational Site Hamburg, Germany, 20246 GSK Investigational Site Koeln, Germany, 50668 GSK Investigational Site Koeln, Germany, 50679 GSK Investigational Site Weimar, Germany, 99427 Collapse << |
NCT03224338 | HIV II Infection | Phase 2 | Recruiting | June 2019 | Portugal ... more >> Centro Hospitalar de Lisboa Central Hospital Curry Cabral Recruiting Lisboa, Portugal Principal Investigator: Fernando Maltez, MD Centro Hospitalar de Lisboa Ocidental Hospital de Egas Moniz Recruiting Lisboa, Portugal Principal Investigator: Kamal Mansinho, MD Centro Hospitalar Lisboa Norte Hospital de Santa Maria Recruiting Lisboa, Portugal Principal Investigator: Nuno Janeiro, MD Hospital Beatriz Ângelo Loures Recruiting Lisboa, Portugal Principal Investigator: Paulo Rodrigues, MD Hospital Garcia de Orta Recruiting Lisboa, Portugal Principal Investigator: Nuno Marques, MD Hospital Professor Doutor Fernando Fonseca Amadora Recruiting Lisboa, Portugal Principal Investigator: Patricia Pacheco, MD Collapse << |
NCT03094507 | HIV | Phase 1 | Completed | - | United Kingdom ... more >> St Stephen's Centre London, United Kingdom, SW10 9NH Collapse << |
NCT02211482 | HIV-1 Infection | Phase 4 | Completed | - | Argentina ... more >> Fundacion Huesped Caba, Buenos Aires, Argentina, C1202ABB Collapse << |
NCT02404805 | HIV Hepatitis... more >> C Collapse << | Not Applicable | Completed | - | United States, Colorado ... more >> University of Colorado Anschutz Medical Campus Aurora, Colorado, United States, 80045 Collapse << |
NCT02976259 | HIV Infection Primary | Phase 3 | Not yet recruiting | January 2020 | - |
NCT01568892 | HIV Infections | Phase 3 | Completed | - | - |
NCT02572947 | Human Immunodeficiency Virus ... more >> Dolutegravir Monotherapy Treatment Efficacy Collapse << | Phase 2 | Completed | - | Switzerland ... more >> University Hospitals of Geneva, HIV unit Geneva, Switzerland, 1205 Collapse << |
NCT01568892 | - | - | Completed | - | - |
NCT02098837 | HIV | Phase 4 | Completed | - | Belgium ... more >> Insititute Of Tropical Medicine Antwerp Antwerp, Belgium, B-2000 CHU Saint-Pierre Brussels, Belgium, 100 Universitaire Ziekenhuis Gent Gent, Belgium, 9000 France Hopital de la Croix Rousse Lyon, France, 69004 Service des Maladies Infectieuses et Tropicales du CHU de NANTES Nantes, France, 44093 Hopital Saint Louis Paris, France, 75010 Pitié-Salpêtrière Hospital Paris, France, 75013 Hospital Bichat Claude-Bernard Paris, France, 75018 Germany Universitätsklinikum Bonn Bonn, Germany, 53127 Universitätsklinikum Essen Essen, Germany, 45147 Klinikum der Goethe-Universität Frankfurt Frankfurt, Germany, 60590 ICH Infektiologisches Centrum Hamburg Hamburg, Germany, 20146 Medizinische Hochschule Hannover Hannover, Germany, 30625 Italy Santa Maria Annunziata di Firenze Firenze, Italy, 50011 San Paolo Hospital Milan, Italy, 20142 Azienda Ospedaliera - Polo Universitario 'Luigi Sacco' Milan, Italy, 20157 Universitaria di Modena Modena, Italy, 41124 Spain Universitario Alicante Alicante, Spain, 03010 Hospital General Universitario de Elche Alicante, Spain, 03203 Hospital de la Santa Creu i Sant Pau Barcelona, Spain, 08025 Hospital Clinic Barcelona Barcelona, Spain, 08036 Universitari de Bellvitge Barcelona, Spain, 08907 IrsiCaixa Barcelona, Spain, 08916 Hospital Ramon y Cajal Madrid, Spain, 28034 Hospital Universitario La Paz Madrid, Spain, 28046 United Kingdom Elton John Centre Brighton, United Kingdom, BN2 1ES Southmead Hospital Bristol, United Kingdom, BS10 5NB Bart's Hospital London, United Kingdom, E1 1BB Royal Free Hospital London, United Kingdom, NW3 2QG St Thomas Hospital London, United Kingdom, SE1 7EH Chelsea & Westminster Hospital London, United Kingdom, Sw10 9NH St Mary's Hospital London, United Kingdom, W2 1NY Mortimer Market Centre London, United Kingdom, WC1E 6JB Collapse << |
NCT02509195 | HIV | Phase 4 | Completed | - | United Kingdom ... more >> St Stephen's Centre, Chelsea & Westminster Hospital London, United Kingdom, SW10 9NH Collapse << |
NCT02500446 | HIV | Phase 4 | Completed | - | Australia, Victoria ... more >> Melbourne Sexual Health Centre Carlton, Victoria, Australia, 3053 Alfred Hospital Prahran, Victoria, Australia, 3010 Collapse << |
NCT02491242 | - | - | Completed | - | Spain ... more >> Ramon y Cajal Hospital Madrid, Spain, 28034 Collapse << |
NCT02924389 | HIV | Not Applicable | Recruiting | June 2020 | United States, Georgia ... more >> Grady Health System Recruiting Atlanta, Georgia, United States, 30303 Contact: Cecile Lahiri, MD 404-616-6306 cdelill@emory.edu Ponce De Leon Center Recruiting Atlanta, Georgia, United States, 30308 Contact: Cecile Lahiri, MD 404-616-6306 cdelill@emory.edu Emory University Recruiting Atlanta, Georgia, United States, 30322 Contact: Cecile Lahiri, MD 404-616-6306 cdelill@emory.edu Collapse << |
NCT02401828 | Human Immunodeficiency Virus | Phase 4 | Active, not recruiting | July 2017 | Netherlands ... more >> Erasmus Medical Center Rotterdam, Zuid Holland, Netherlands, 3000 CA Collapse << |
NCT03016533 | HIV Infections | Phase 3 | Recruiting | December 29, 2023 | South Africa ... more >> GSK Investigational Site Recruiting Hillbrow, Gauteng, South Africa, 2001 Contact: US GSK Clinical Trials Call Center 877-379-3718 GSKClinicalSupportHD@gsk.com Contact: EU GSK Clinical Trials Call Center +44 (0) 20 8990 4466 GSKClinicalSupportHD@gsk.com Thailand GSK Investigational Site Recruiting Chiang Mai, Thailand, 50200 Contact: US GSK Clinical Trials Call Center 877-379-3718 GSKClinicalSupportHD@gsk.com Contact: EU GSK Clinical Trials Call Center +44 (0) 20 8990 4466 GSKClinicalSupportHD@gsk.com Collapse << |
NCT02487706 | HIV | Phase 4 | Completed | - | Spain ... more >> Germans Trias i Pujol Hospital Badalona, Barcelona, Spain, 08916 Collapse << |
NCT02566707 | HIV-1 Infection | Phase 2 | Terminated(due to introduction... more >> of another integrase inhibitor, recruitement was not feasible anymore.) Collapse << | - | Germany ... more >> University of Bonn Bonn, Germany Netherlands Rijstate Arnhem, Netherlands Radboud University Nijmegen Medical Centre Nijmegen, Netherlands St. Elisabeth Tilburg, Netherlands Collapse << |
靶点 | Description | IC50 |
---|---|---|
HIV Integrase | IC50:2.7nM |
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